Assay Report Card

Basic Information

ID: ALA4670933

Type: Binding

Description: Potency index, ratio of afatinib Kinact to test compound Kinact for inhibition of C-terminal His6-tagged HER2-A775_G776insYVMA mutant (703 to 1029 residues) (unknown origin) expressed in Sf9 insect cells

Organism: Homo sapiens

Cell type: Sf9

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
545.605.265.26
584.086.066.06
496.966.126.12
514.555.295.29