Assay Report Card

Basic Information

ID: ALA4673853

Type: Binding

Description: Competitive inhibition of recombinant SETD8 catalytic domain (unknown origin) (232 to 393 residues) expressed in Escherichia coli using biotinylated H4 (1 to 24) peptide substrate measured after 15 mins in presence of varying levels of [3H-SAM] by scintillation counting assay

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
442.613.253.25