Assay Report Card

Basic Information

ID: ALA4673854

Type: Binding

Description: Competitive inhibition of recombinant SETD8 catalytic domain (unknown origin) (232 to 393 residues) expressed in Escherichia coli using varying levels of biotinylated H4 (1 to 24) peptide substrate measured after 15 mins in presence of [3H-SAM] by scintillation counting assay

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
442.613.253.25