Basic Information
ID: ALA4673856
Type: Binding
Description: Inhibition of recombinant SETD8 catalytic domain (unknown origin) (232 to 393 residues) expressed in Escherichia coli assessed as reduction in incorporation of [3H]-labeled methyl group into biotinylated H4 (1 to 24) peptide measured after 1 hr using [3H-SAM] by scintillation proximity assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4673856
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 399.50 | 2.38 | 2.38 |
| 385.47 | 2.35 | 2.35 |
| 442.61 | 3.25 | 3.25 |