Assay Report Card

Basic Information

ID: ALA4675813

Type: ADME

Description: Inhibition of recombinant human GST-tagged JAK2 catalytic domain (809 to 1153+9 residues) expressed in baculovirus expression system using FITC-KGGEEEEYFELVKK as substrate in presence of ATP at Km by microfluidic assay

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
383.422.542.54
387.451.941.94
383.422.542.54
369.392.532.53
398.431.441.44
369.392.532.53
383.422.542.54
388.442.412.41
401.431.461.46
413.492.332.33
388.442.412.41
383.422.542.54
441.422.482.48
397.452.932.93
397.452.932.93
369.392.532.53
403.450.910.91
369.392.532.53