Assay Report Card

Basic Information

ID: ALA4677816

Type: Binding

Description: Inhibition of human FGFR4 assessed as remaining enzyme activity at 0.2 uM using poly (Glu, Tyr)4:1 as substrate incubated for 20 mins followed by [33P]-ATP addition and measured after 120 mins by radiometric hotspot assay relative to control

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
509.396.806.80
476.582.712.71
454.494.524.52
463.583.483.48
450.542.492.49
450.542.492.49
478.534.444.44
286.292.342.34
500.632.642.64
451.531.881.88
442.484.684.68
456.504.694.69
448.523.843.84
456.504.994.99
416.443.913.91