ID: ALA4680578
Type: Binding
Description: Inhibition of recombinant His-tagged human G9a expressed in Escherichia coli BL21 (DE3) using biotin-labeled histone H3-20 peptide as substrate incubated for 30 mins in presence of [3H]-SAM cofactor by scintillation proximity assay
Format: BAO_0000019
Organism: Homo sapiens
Target: Histone-lysine N-methyltransferase, H3 lysine-9 specific 3(ALA6032)
Document: ALA4680065
Inhibition of recombinant His-tagged human G9a expressed in Escherichia coli BL21 (DE3) using biotin-labeled histone H3-20 peptide as substrate incubated for 30 mins in presence of [3H]-SAM cofactor by scintillation proximity assay: 1
Bioactivity
Activity Types for Assay ALA4680578
IC50
Parent Molecular Weight | ALogP | Polar Surface Area |
---|---|---|
368.44 | 4.15 | 4.15 |
392.47 | 2.52 | 2.52 |
382.42 | 0.25 | 0.25 |
369.43 | 3.28 | 3.28 |
262.28 | 1.89 | 1.89 |