Basic Information
ID: ALA4680578
Type: Binding
Description: Inhibition of recombinant His-tagged human G9a expressed in Escherichia coli BL21 (DE3) using biotin-labeled histone H3-20 peptide as substrate incubated for 30 mins in presence of [3H]-SAM cofactor by scintillation proximity assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4680578
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 368.44 | 4.15 | 4.15 |
| 392.47 | 2.52 | 2.52 |
| 382.42 | 0.25 | 0.25 |
| 369.43 | 3.28 | 3.28 |
| 262.28 | 1.89 | 1.89 |