Basic Information
ID: ALA4682087
Type: Binding
Description: Activation of human GABAB1/GABAB2 expressed in HEK293 cells co-transfected with rat CaV2.2 channel assessed as reduction in CaV2.2-mediated peak-current amplitude in response to the depolarizing pulse by whole cell patch clamp assay
Organism: Homo sapiens
Cell type: HEK293T
Activity Charts
Bioactivity
Activity Types for Assay ALA4682087
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 1796.07 | ||
| 1825.12 | ||
| 1811.04 | ||
| 1895.16 | ||
| 1957.23 | ||
| 1894.23 | ||
| 1852.14 | ||
| 1853.13 | ||
| 1915.15 |