Basic Information
ID: ALA4682088
Type: Binding
Description: Selectivity index, ratio of IC50 for inhibition of human alpha9alpha10 nAChR expressed in Xenopus laevis oocytes to IC50 for activation of human GABAB1/GABAB2 expressed in HEK293 cells co-transfected with rat CaV2.2 channel assessed as reduction in CaV2.2-mediated peak-current amplitude
Activity Charts
Bioactivity
Activity Types for Assay ALA4682088
Ratio IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 1811.04 | ||
| 1957.23 | ||
| 1853.13 | ||
| 1915.15 |