Assay Report Card

Basic Information

ID: ALA4682101

Type: Binding

Description: Activation of human GABAB1/GABAB2 expressed in HEK293 cells co-transfected with rat CaV2.2 channel assessed as reduction in CaV2.2-mediated Ba2+ peak-current amplitude in response to depolarizing pulse in presence of 1 uM GABAB receptor antagonist CGP55845 by whole cell patch clamp assay

Organism: Homo sapiens

Cell type: HEK293T

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
1811.04
1957.23
1853.13