Assay Report Card

Basic Information

ID: ALA4682104

Type: Binding

Description: Selectivity index, ratio of IC50 for inhibition of rat alpha9alpha10 nAChR expressed in Xenopus laevis oocytes to IC50 for activation of human GABAB1/GABAB2 expressed in HEK293 cells co-transfected with rat CaV2.2 channel assessed as reduction in CaV2.2-mediated peak Ba2+ current amplitude

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
1811.04
1895.16
1957.23
1852.14
1853.13