Basic Information
ID: ALA4683211
Type: Binding
Description: Allosteric inhibition of IKKbeta (unknown origin) using 5FAM-GRHDSGLDSMK-NH2 as substrate pretreated for 10 mins followed measured after 2 hrs by TR-FRET assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4683211
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 592.16 | 7.17 | 7.17 |
| 587.74 | 6.52 | 6.52 |
| 602.71 | 6.42 | 6.42 |
| 636.61 | 7.28 | 7.28 |
| 575.71 | 6.66 | 6.66 |
| 571.74 | 6.82 | 6.82 |
| 636.61 | 7.28 | 7.28 |
| 572.73 | 6.10 | 6.10 |
| 587.74 | 6.52 | 6.52 |
| 572.73 | 6.10 | 6.10 |
| 571.74 | 6.82 | 6.82 |
| 592.16 | 7.17 | 7.17 |
| 614.77 | 6.47 | 6.47 |
| 575.71 | 6.66 | 6.66 |
| 582.73 | 6.39 | 6.39 |
| 547.65 | 5.88 | 5.88 |
| 554.67 | 5.61 | 5.61 |