Assay Report Card

Basic Information

ID: ALA4685798

Type: Binding

Description: Inhibition of chymotrypsin-like activity of human 20S proteasome beta5 subunit at 50 uM using Suc-LLVY-Glo as substrate incubated for 2 hrs followed by substrate addition and measured for 10 mins by bioluminescent assay relative to control

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
576.722.322.32
461.654.064.06
563.653.663.66
533.634.044.04
645.784.324.32
639.754.784.78
529.633.643.64
611.703.563.56
529.633.263.26
606.741.941.94
644.175.915.91
654.724.684.68
620.772.332.33
590.742.712.71
688.625.535.53
623.755.085.08
590.742.712.71
626.155.225.22
499.613.633.63
620.772.332.33
641.723.673.67
559.663.273.27
640.185.525.52
627.703.273.27
533.633.173.17
675.804.334.33