Assay Report Card

Basic Information

ID: ALA4685803

Type: Binding

Description: Reversible inhibition of human 20S proteasome beta5 subunit assessed as residual enzyme activity using Suc-LLVY-Glo as substrate preincubated for 2 hrs followed by compound washout and further incubated for 4 hrs followed by substrate addition and measured after 10 mins by bioluminescent assay relative to control

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
384.25
461.654.064.06
620.772.332.33
342.420.890.89