Assay Report Card

Basic Information

ID: ALA4688541

Type: Binding

Description: Antagonist activity at human histamine 3 receptor transfected in human HEK293T cells assessed as reduction in histamine-induced activity at 10 uM incubated for 30 mins followed by histamine stimulation and measured immediately by BRET assay

Organism: Homo sapiens

Cell type: HEK293T

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
288.391.801.80
334.463.463.46
294.402.562.56
314.473.093.09
350.514.114.11
308.432.902.90