Basic Information
ID: ALA4700949
Type: Unassigned
Description: Ratio of EC50 for activation of human NPFF2R overexpressing CHO cells assessed as inhibition of forskolin-stimulated cAMP degradation incubated for 30 mins in presence of IBMX and 10% FBS by fluorescence based assay to EC50 for activation of human GPR10 overexpressed in CHO-K1 cells assessed as increase in beta arrestin recruitment incubated for 90 mins by PathHunter assay
Format: BAO_0000219
Target: Unchecked(ALA612545)
Document: ALA4699444
Ratio of EC50 for activation of human NPFF2R overexpressing CHO cells assessed as inhibition of forskolin-stimulated cAMP degradation incubated for 30 mins in presence of IBMX and 10% FBS by fluorescence based assay to EC50 for activation of human GPR10 overexpressed in CHO-K1 cells assessed as increase in beta arrestin recruitment incubated for 90 mins by PathHunter assay: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4700949
Ratio EC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 4489.22 | ||
| 4274.02 | ||
| 4330.12 | ||
| 4244.97 | ||
| 4302.07 | ||
| 3730.27 | ||
| 4545.33 | ||
| 4517.27 | ||
| 4358.09 |