Basic Information
ID: ALA4701012
Type: Functional
Description: Antagonist activity at human adenosine 2A receptor expressed in T-REx-CHO cells preincubated for 1 hr followed by NECA stimulation and measured after 30 mins by Eu-cAMP tracer based TR-FRET assay
Format: BAO_0000219
Organism: Homo sapiens
Cell type: T-REX-CHO
Target: Adenosine A2a receptor(ALA251)
Document: ALA4699449
Antagonist activity at human adenosine 2A receptor expressed in T-REx-CHO cells preincubated for 1 hr followed by NECA stimulation and measured after 30 mins by Eu-cAMP tracer based TR-FRET assay: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4701012
Kb
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 363.38 | 2.17 | 2.17 |
| 461.40 | 1.93 | 1.93 |
| 391.44 | 2.15 | 2.15 |