Competitive orthosteric antagonist activity at human GPR7 expressed in CHO cell membranes assessed as increase in Koff rate kinetics of [125I]-labeled...

Basic Information

ID: ALA4701820

Type: Binding

Description: Competitive orthosteric antagonist activity at human GPR7 expressed in CHO cell membranes assessed as increase in Koff rate kinetics of [125I]-labeled human NPW23 at 0 to 30 uM by real-time scintillation proximity binding assay

Format: BAO_0000249

Organism: Homo sapiens

Cell type: CHO

Subcellular Fraction: Cell membrane

Target:  Neuropeptides B/W receptor type 1(ALA1293293)

Document:  ALA4699486

Competitive orthosteric antagonist activity at human GPR7 expressed in CHO cell membranes assessed as increase in Koff rate kinetics of [125I]-labeled human NPW23 at 0 to 30 uM by real-time scintillation proximity binding assay: 1

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
397.195.955.95