Assay Report Card

Basic Information

ID: ALA4705027

Type: Binding

Description: Selectivity ratio of IC50 for human PNMT C183A mutant using PEA as substrate and AdoMet as co-substrate to IC50 for inhibition of C-terminal hexahistidine tag in human recombinant PNMT expressed in Escherichia coli assessed as inhibitor dissociation constant in presence of 5 uM PEA as substrate and AdoMet as co-substrate

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
326.38-1.28-1.28