Basic Information
ID: ALA4705251
Type: Binding
Description: Agonist activity at EA-fragment beta-arrestin-tagged human MOR/DOR expressed in human U2OS cell membranes assessed as stimulation beta-arrestin recruitment at 10 uM after 60 mins by Pathhunter chemiluminescence assay relative to DAMGO
Organism: Homo sapiens
Cell type: U2OS
Subcellular Fraction: Cell membrane
Activity Charts
Bioactivity
Activity Types for Assay ALA4705251
Emax
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 782.90 | -1.27 | -1.27 |
| 408.54 | 4.42 | 4.42 |
| 500.64 | 4.54 | 4.54 |
| 505.68 | 5.21 | 5.21 |
| 489.62 | 4.74 | 4.74 |
| 550.12 | 5.65 | 5.65 |
| 469.63 | 4.82 | 4.82 |
| 475.68 | 5.35 | 5.35 |
| 501.65 | 5.00 | 5.00 |
| 529.70 | 5.04 | 5.04 |
| 529.70 | 5.31 | 5.31 |
| 485.63 | 5.15 | 5.15 |
| 505.63 | 4.59 | 4.59 |
| 549.69 | 5.91 | 5.91 |
| 516.66 | 4.40 | 4.40 |
| 521.70 | 5.06 | 5.06 |
| 499.66 | 5.15 | 5.15 |
| 516.66 | 4.40 | 4.40 |
| 515.67 | 5.00 | 5.00 |