Basic Information
ID: ALA4709469
Type: Binding
Description: Inhibition of full length recombinant human N-terminal GST/His6-tagged PAK4 expressed in baculovirus infected sf9 insect cells using tetra LRRWSLG as substrate preincubated for 20 min followed by [gamma33P]ATP addition and measured after 120 mins by Hotspot assay
Format: BAO_0000219
Organism: Homo sapiens
Cell type: Sf9
Target: Serine/threonine-protein kinase PAK 4(ALA4482)
Document: ALA4706541
Inhibition of full length recombinant human N-terminal GST/His6-tagged PAK4 expressed in baculovirus infected sf9 insect cells using tetra LRRWSLG as substrate preincubated for 20 min followed by [gamma33P]ATP addition and measured after 120 mins by Hotspot assay: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4709469
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 490.64 | 4.53 | 4.53 |
| 392.85 | 3.70 | 3.70 |
| 406.87 | 4.09 | 4.09 |
| 469.93 | 4.67 | 4.67 |
| 432.91 | 4.48 | 4.48 |
| 476.96 | 4.50 | 4.50 |