Basic Information
ID: ALA4709494
Type: Binding
Description: Inhibition of full length recombinant human N-terminal GST/His6-tagged PAK1 expressed in sf9 insect cells assessed as residual activity at 0.1 uM using tetra LRRWSLG as substrate preincubated for 20 min followed by [gamma33P]ATP addition and measured after 120 mins by Hotspot assay relative to control
Format: BAO_0000219
Organism: Homo sapiens
Cell type: Sf9
Target: Serine/threonine-protein kinase PAK 1(ALA4600)
Document: ALA4706541
Inhibition of full length recombinant human N-terminal GST/His6-tagged PAK1 expressed in sf9 insect cells assessed as residual activity at 0.1 uM using tetra LRRWSLG as substrate preincubated for 20 min followed by [gamma33P]ATP addition and measured after 120 mins by Hotspot assay relative to control: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4709494
Activity
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 469.93 | 4.67 | 4.67 |