Basic Information
ID: ALA4709751
Type: Binding
Description: Inhibition of recombinant full length His-tagged human CDK9/cyclin T1 expressed in baculovirus expression system using biotinylated peptide biotin-Ttds-YISPLKSPYKISEG as substrate preincubated for 15 mins followed by ATP and substrate addition and measured after 25 mins by TR-FRET assay
Format: BAO_0000019
Organism: Homo sapiens
Target: CDK9/cyclin T1(ALA2111389)
Document: ALA4706546
Inhibition of recombinant full length His-tagged human CDK9/cyclin T1 expressed in baculovirus expression system using biotinylated peptide biotin-Ttds-YISPLKSPYKISEG as substrate preincubated for 15 mins followed by ATP and substrate addition and measured after 25 mins by TR-FRET assay: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4709751
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 422.43 | 4.49 | 4.49 |
| 387.44 | 3.61 | 3.61 |
| 388.42 | 2.97 | 2.97 |
| 389.41 | 2.22 | 2.22 |
| 404.44 | 4.35 | 4.35 |
| 421.45 | 5.12 | 5.12 |