ID: ALA4711941
Type: Functional
Description: Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15 mins followed by WO459 addition and measured after 30 mins by LANCE Ultra cAMP kit based microplate reader analysis
Organism: Homo sapiens
Cell type: HEK293
Bioactivity
Activity Types for Assay ALA4711941
IC50
Parent Molecular Weight | ALogP | Polar Surface Area |
---|---|---|
264.37 | 4.38 | 4.38 |
236.31 | 4.06 | 4.06 |
250.34 | 4.37 | 4.37 |
312.41 | 5.73 | 5.73 |
254.30 | 4.20 | 4.20 |
237.30 | 3.45 | 3.45 |
250.34 | 4.37 | 4.37 |
315.21 | 4.82 | 4.82 |
243.35 | 3.19 | 3.19 |
286.37 | 5.21 | 5.21 |
312.41 | 5.73 | 5.73 |
250.34 | 4.37 | 4.37 |
315.21 | 4.82 | 4.82 |
266.34 | 4.07 | 4.07 |
264.37 | 4.68 | 4.68 |
160.22 | 2.84 | 2.84 |
286.37 | 5.21 | 5.21 |
226.28 | 3.65 | 3.65 |
242.34 | 4.12 | 4.12 |
240.31 | 2.79 | 2.79 |
254.30 | 4.20 | 4.20 |
226.28 | 3.65 | 3.65 |
237.30 | 3.45 | 3.45 |
237.30 | 3.45 | 3.45 |
266.34 | 4.07 | 4.07 |
254.30 | 4.20 | 4.20 |
242.34 | 4.12 | 4.12 |
266.34 | 4.07 | 4.07 |
312.41 | 5.73 | 5.73 |