Basic Information
ID: ALA4712180
Type: Functional
Description: Antagonist activity at recombinant human N-terminal epitope tagged/eYFP-fused FLAG-tagged GPR84 expressed in Flp-In TREx 293 cells assessed as inhibition of embelin-induced [35S]GTPgammaS binding pre-incubated for 15 mins followed by [35S]GTPgammaS addition and measured after 45 mins by liquid scintillation spectrometry
Organism: Homo sapiens
Cell type: Flp-In-T-REx-293
Activity Charts
Bioactivity
Activity Types for Assay ALA4712180
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 452.47 | 2.10 | 2.10 |
| 442.51 | 2.20 | 2.20 |
| 443.50 | 2.72 | 2.72 |