Basic Information
ID: ALA4717253
Type: Binding
Description: Antagonist activity at human full-length MCR assessed as inhibition of receptor binding to co-activator peptide by PathHunter assay
Format: BAO_0000357
Organism: Homo sapiens
Target: Mineralocorticoid receptor(ALA1994)
Document: ALA4715716
Antagonist activity at human full-length MCR assessed as inhibition of receptor binding to co-activator peptide by PathHunter assay: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4717253
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 416.58 | 4.85 | 4.85 |
| 414.50 | 3.12 | 3.12 |
| 392.91 | 3.81 | 3.81 |
| 419.93 | 3.57 | 3.57 |
| 410.85 | 3.57 | 3.57 |
| 342.76 | 4.07 | 4.07 |
| 358.42 | 2.78 | 2.78 |
| 468.96 | 5.10 | 5.10 |
| 392.86 | 3.43 | 3.43 |
| 420.92 | 3.99 | 3.99 |
| 352.19 | 4.85 | 4.85 |
| 482.99 | 4.83 | 4.83 |
| 335.74 | 4.34 | 4.34 |
| 464.82 | 4.46 | 4.46 |
| 446.96 | 4.38 | 4.38 |
| 436.92 | 3.23 | 3.23 |
| 428.77 | 4.70 | 4.70 |
| 470.98 | 5.13 | 5.13 |
| 487.93 | 4.50 | 4.50 |
| 431.90 | 3.50 | 3.50 |
| 317.75 | 4.20 | 4.20 |
| 376.41 | 2.91 | 2.91 |
| 406.89 | 3.60 | 3.60 |
| 507.02 | 5.92 | 5.92 |
| 420.92 | 3.99 | 3.99 |
| 388.45 | 2.78 | 2.78 |
| 420.92 | 3.99 | 3.99 |
| 462.02 | 4.73 | 4.73 |
| 427.31 | 4.08 | 4.08 |
| 389.81 | 4.37 | 4.37 |