Basic Information
ID: ALA4718883
Type: Binding
Description: Inhibition of recombinant human His-tagged PRKACA (1 to 351 residues) expressed in Escherichia coli expression system at 500 nM using Ser/Thr 01 as substrate incubated for 1 hr in presence of ATP at its Km concentration by Z'-LYTE assay relative to control
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4718883
Inhibition
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 393.44 | 3.41 | 3.41 |
| 448.55 | 3.56 | 3.56 |
| 374.44 | 4.17 | 4.17 |
| 330.39 | 3.77 | 3.77 |
| 360.42 | 3.78 | 3.78 |
| 344.42 | 4.16 | 4.16 |