Assay Report Card

Basic Information

ID: ALA4718895

Type: Binding

Description: Inhibition of human LAT1 expressed in HEK293-T-Rex cells assessed as inhibition of [3H]-gabapentin uptake at 200 uM by scintillation counting cis-inhibition assay

Organism: Homo sapiens

Cell type: HEK293-T-REx

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
75.07-0.97-0.97
181.190.350.35
165.190.640.64
131.170.440.44
204.231.121.12
180.210.060.06
90.08-1.55-1.55
196.21-0.23-0.23
174.20-1.34-1.34
219.240.540.54
182.65-0.13-0.13
242.30-0.37-0.37
258.30-0.66-0.66
189.220.440.44