Assay Report Card

Basic Information

ID: ALA4722344

Type: Functional

Description: Allosteric antagonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as inhibition of UTP-induced intracellular calcium influx at 3 to 10 uM preincubated for 20 mins followed by UTP addition measured at 0.4 secs interval for 60 times by Oregon Green BAPTA-1/AM dye-based fluorescence assay

Organism: Homo sapiens

Cell type: 1321N1

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
432.844.274.27