Basic Information
ID: ALA4724701
Type: Binding
Description: Ratio of IC50 for protac activity at NanoLuc-tagged VHL/ERK5 in HEK293 cells assessed as inhibition of VHL activity incubated for 2 hrs by NanoBRET live cell assay to IC50 for protac activity at VHL/ERK5 (unknown origin) assessed as inhibition of VHK activity by measuring phosphorylated
Format: BAO_0000219
Organism: Homo sapiens
Target: Unchecked(ALA612545)
Document: ALA4715905
Ratio of IC50 for protac activity at NanoLuc-tagged VHL/ERK5 in HEK293 cells assessed as inhibition of VHL activity incubated for 2 hrs by NanoBRET live cell assay to IC50 for protac activity at VHL/ERK5 (unknown origin) assessed as inhibition of VHK activity by measuring phosphorylated: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4724701
Ratio IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 1034.13 |