Assay Report Card

Basic Information

ID: ALA4724701

Type: Binding

Description: Ratio of IC50 for protac activity at NanoLuc-tagged VHL/ERK5 in HEK293 cells assessed as inhibition of VHL activity incubated for 2 hrs by NanoBRET live cell assay to IC50 for protac activity at VHL/ERK5 (unknown origin) assessed as inhibition of VHK activity by measuring phosphorylated

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
1034.13