Assay Report Card

Basic Information

ID: ALA4726639

Type: Binding

Description: Protac activity at VHL/ERalpha in human MCF7 cells assessed as induction of ERalpha protein degradation by measuring ERalpha protein level at 20 uM incubated for 8 hrs in presence of proteasome inhibitor, MG132 by western blot analysis relative to lamin B

Organism: Homo sapiens

Cell type: MCF7

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
3094.84