Inhibition of recombinant human CDC7/Dbf4 expressed in baculovirus infected Sf9 insect cells assessed as inhibition of fluorescein labelled substrate ...

Basic Information

ID: ALA4734043

Type: Binding

Description: Inhibition of recombinant human CDC7/Dbf4 expressed in baculovirus infected Sf9 insect cells assessed as inhibition of fluorescein labelled substrate phosphorylation in presence of ATP at 10 uM measured after 60 mins by TR-FRET assay

Format: BAO_0000219

Organism: Homo sapiens

Cell type: Sf9

Target:  CDC7/DBF4 (Cell division cycle 7-related protein kinase/Activator of S phase kinase)(ALA2111377)

Document:  ALA4732086

Inhibition of recombinant human CDC7/Dbf4 expressed in baculovirus infected Sf9 insect cells assessed as inhibition of fluorescein labelled substrate phosphorylation in presence of ATP at 10 uM measured after 60 mins by TR-FRET assay: 1

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
258.373.983.98
584.225.385.38
332.434.174.17
401.325.475.47
415.355.525.52
415.355.525.52
468.436.206.20
337.274.754.75
401.325.475.47
415.355.525.52
382.444.494.49