Assay Report Card

Basic Information

ID: ALA4739794

Type: Binding

Description: Inhibition of biotinylated-THZ1 binding to CDK12/CDK13 in human Jurkat cells assessed as reduction in cyclin K pull down at 500 nM preincubated for 4 hrs followed by biotinylated-THZ1 addition by Western blotting based pulldown assay

Organism: Homo sapiens

Cell type: Jurkat

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
539.735.875.87
555.735.575.57
525.705.565.56
511.675.175.17