Assay Report Card

Basic Information

ID: ALA4739798

Type: Binding

Description: Inhibition of biotinylated-THZ1 binding to CDK12 in human Jurkat cells assessed as reduction in cyclin K pull down at 1 uM preincubated for 6 hrs followed by biotinylated-THZ1 addition by Western blotting based pull-down assay

Organism: Homo sapiens

Cell type: Jurkat

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
472.985.485.48
473.974.884.88
531.064.814.81
545.096.146.14
487.996.206.20
559.074.454.45