ID: ALA4742444
Type: Binding
Description: Inhibition of kinase tracer 236 binding to full-length His-tagged recombinant human CDK8/cyclin C incubated for 60 mins by FRET based LanthaScreen Eu-Kinase binding assay
Organism: Homo sapiens
Bioactivity
Activity Types for Assay ALA4742444
IC50
Parent Molecular Weight | ALogP | Polar Surface Area |
---|---|---|
395.43 | 3.92 | 3.92 |
297.36 | 2.74 | 2.74 |
387.36 | 4.49 | 4.49 |
415.42 | 4.98 | 4.98 |
327.38 | 2.53 | 2.53 |
311.39 | 3.22 | 3.22 |
297.36 | 3.19 | 3.19 |
297.36 | 3.19 | 3.19 |
329.38 | 3.17 | 3.17 |
335.36 | 3.18 | 3.18 |
299.33 | 2.04 | 2.04 |
269.30 | 1.96 | 1.96 |
313.36 | 2.07 | 2.07 |
347.85 | 3.22 | 3.22 |
394.40 | 2.91 | 2.91 |
345.83 | 3.87 | 3.87 |
326.36 | 1.41 | 1.41 |
283.33 | 2.44 | 2.44 |
349.39 | 3.48 | 3.48 |
349.39 | 3.48 | 3.48 |
377.44 | 3.97 | 3.97 |
301.32 | 2.39 | 2.39 |
441.48 | 4.52 | 4.52 |
377.44 | 3.97 | 3.97 |
343.38 | 1.69 | 1.69 |
283.33 | 2.68 | 2.68 |
359.39 | 3.35 | 3.35 |
347.80 | 2.72 | 2.72 |
325.41 | 3.68 | 3.68 |
299.33 | 1.58 | 1.58 |
331.35 | 2.02 | 2.02 |
311.39 | 3.17 | 3.17 |