Basic Information
ID: ALA4767588
Type: Binding
Description: Inhibition of mouse GAT4 expressed in HEK293 cell line assessed as inhibition of [3H]GABA uptake measured after 35 mins by liquid scintillation method
Organism: Mus musculus
Cell type: HEK293
Activity Charts
Bioactivity
Activity Types for Assay ALA4767588
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 505.61 | 4.82 | 4.82 |
| 350.42 | 3.17 | 3.17 |
| 519.64 | 5.13 | 5.13 |
| 419.31 | 4.73 | 4.73 |
| 468.69 | 5.17 | 5.17 |
| 500.71 | 5.78 | 5.78 |
| 517.16 | 6.29 | 6.29 |
| 500.71 | 5.43 | 5.43 |
| 454.66 | 4.86 | 4.86 |
| 482.72 | 5.81 | 5.81 |
| 502.15 | 5.87 | 5.87 |
| 544.19 | 6.04 | 6.04 |
| 448.65 | 3.79 | 3.79 |
| 503.13 | 5.90 | 5.90 |
| 502.15 | 5.87 | 5.87 |
| 482.72 | 5.56 | 5.56 |
| 414.60 | 5.43 | 5.43 |
| 489.11 | 5.51 | 5.51 |
| 472.65 | 5.00 | 5.00 |
| 517.16 | 6.29 | 6.29 |
| 496.74 | 5.94 | 5.94 |
| 522.66 | 5.88 | 5.88 |
| 486.68 | 5.39 | 5.39 |
| 467.70 | 5.21 | 5.21 |
| 504.67 | 5.53 | 5.53 |
| 482.72 | 5.64 | 5.64 |
| 503.13 | 5.90 | 5.90 |
| 468.69 | 5.25 | 5.25 |
| 489.11 | 5.51 | 5.51 |
| 481.73 | 5.52 | 5.52 |
| 105.09 | -1.61 | -1.61 |
| 485.69 | 5.35 | 5.35 |