Assay Report Card

Basic Information

ID: ALA4769546

Type: ADME

Description: Inhibition of GST-tagged human recombinant PI3Kgamma catalytic domain (468 to 1203 residues) expressed in insect cells using PIP2 peptide as substrate incubated for 1 hr in presence ATP by ADP-Glo Kinase Assay

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
380.412.922.92
441.483.843.84
514.573.773.77
489.544.694.69
488.533.663.66
489.544.694.69
505.995.215.21
499.563.463.46