Assay Report Card

Basic Information

ID: ALA4771346

Type: Functional

Description: In vivo inhibition of STAT3 in BALB/c mouse xenografted with human MDA-MB-231 cells assessed as reduction in STAT3 Y705 phosphorylation in tumor tissue at 10 mg/kg, ip administered once daily for 21 days and measured on day 21 by immunofluorescent staining based fluorescence microscopy

Organism: Mus musculus

Strain: BALB/c

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
311.292.872.87