Assay Report Card

Basic Information

ID: ALA4772592

Type: Binding

Description: Inverse agonist activity at human RORgammat assessed as inhibition of N-terminal biotinylated co-activator SRC1 recruitment measured after 60 mins by FRET assay

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
532.376.536.53
515.325.915.91
527.336.826.82
548.376.376.37
527.336.826.82
549.287.067.06
533.366.286.28
546.407.317.31
481.384.874.87
547.386.676.67
472.465.825.82
547.747.167.16
528.316.466.46
532.376.286.28
519.377.077.07
360.414.304.30
455.464.924.92
506.916.726.72
509.346.776.77
576.385.575.57
548.376.256.25
529.306.006.00
513.306.516.51
499.276.586.58
531.296.986.98
529.306.346.34
514.295.905.90
548.375.795.79
527.336.906.90
534.345.535.53
576.385.715.71
517.896.296.29
527.337.077.07
492.886.426.42
519.376.976.97
531.296.656.65
518.387.017.01
531.296.656.65