Assay Report Card

Basic Information

ID: ALA4775171

Type: Functional

Description: Antagonist activity at human MC4R expressed in HEK293 cells expressing the GScAMP22F cAMP reporter assessed as reduction in alpha-MSH-induced cAMP accumulation by cAMP split-luciferase reporter gene assay

Organism: Homo sapiens

Cell type: HEK293

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
1074.26
1075.25
1108.70
1110.33
1050.23
1158.33
1110.33
1088.32
1092.25
1034.23
1075.25
1098.28
1108.70
1098.28
1092.25
1122.30
1114.32
1092.25
1108.27
1088.29
1108.70