Basic Information
ID: ALA4775347
Type: Binding
Description: Displacement of [125I] [NIe75, Tyr77]Pyr-apelin-13 from YFP-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr by gamma counting based Cheng-Prusoff equation analysis
Format: BAO_0000219
Organism: Homo sapiens
Cell type: HEK293
Target: Apelin receptor(ALA1628481)
Document: ALA4765470
Displacement of [125I] [NIe75, Tyr77]Pyr-apelin-13 from YFP-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr by gamma counting based Cheng-Prusoff equation analysis: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4775347
Ki
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 1533.83 | ||
| 1053.28 | ||
| 1176.43 | ||
| 1171.41 | ||
| 838.97 | -2.56 | -2.56 |
| 1212.46 | ||
| 1162.40 | ||
| 1222.50 | ||
| 1212.46 | ||
| 1180.44 | ||
| 1169.40 | ||
| 1318.59 | ||
| 1707.07 | ||
| 1065.29 | ||
| 1262.53 | ||
| 1176.43 | ||
| 1136.37 | ||
| 1266.51 | ||
| 1049.24 | ||
| 1125.38 | ||
| 1268.53 | ||
| 1212.46 | ||
| 1051.26 | ||
| 1238.50 | ||
| 1162.40 | ||
| 1178.40 | ||
| 1196.42 | ||
| 1051.26 | ||
| 1162.40 | ||
| 1174.42 | ||
| 1115.35 | ||
| 1222.50 | ||
| 1178.47 | ||
| 1162.40 | ||
| 1178.45 | ||
| 1096.34 | ||
| 1216.50 | ||
| 1162.40 | ||
| 1202.47 | ||
| 1093.34 | ||
| 1065.29 | ||
| 1176.43 | ||
| 1176.43 | ||
| 1132.33 | ||
| 1086.31 | ||
| 1139.41 | ||
| 1147.39 | ||
| 1176.43 | ||
| 1210.45 | ||
| 1146.36 | ||
| 1262.53 | ||
| 1168.45 | ||
| 1210.45 | ||
| 1079.31 | ||
| 1134.35 | ||
| 1178.49 | ||
| 1224.48 | ||
| 3865.71 | ||
| 1252.53 | ||
| 1216.50 | ||
| 1023.21 | ||
| 1148.38 | ||
| 1160.39 | ||
| 1162.40 | ||
| 1268.53 | ||
| 1172.44 | ||
| 1179.46 | ||
| 952.13 | -2.03 | -2.03 |
| 1017.24 | ||
| 1079.31 | ||
| 1211.48 |