Basic Information
ID: ALA4775349
Type: Functional
Description: Agonist activity at human APJ receptor expressed in HEK293T cells co-expressing PDZ-Rho-Gef-RLucll assessed as induction of Galpha12 effector (PDZ-RhoGEF) to the cell membrane incubated for 5 mins by BRET assay
Format: BAO_0000219
Organism: Homo sapiens
Cell type: HEK293T
Target: Apelin receptor(ALA1628481)
Document: ALA4765470
Agonist activity at human APJ receptor expressed in HEK293T cells co-expressing PDZ-Rho-Gef-RLucll assessed as induction of Galpha12 effector (PDZ-RhoGEF) to the cell membrane incubated for 5 mins by BRET assay: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4775349
EC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 1533.83 | ||
| 1212.46 | ||
| 1212.46 | ||
| 1180.44 | ||
| 1318.59 | ||
| 1262.53 | ||
| 1212.46 | ||
| 1162.40 | ||
| 1162.40 | ||
| 1178.45 | ||
| 1162.40 | ||
| 1202.47 | ||
| 1093.34 | ||
| 1176.43 | ||
| 1176.43 | ||
| 1210.45 | ||
| 1262.53 | ||
| 1168.45 | ||
| 1210.45 | ||
| 1079.31 | ||
| 3865.71 | ||
| 1216.50 | ||
| 1160.39 |