Displacement of [3H]ZM2421385 from adenosine A2A receptor expressed in human HeLa cell membranes at 1 uM incubated for 30 mins by scintillation counti...

Basic Information

ID: ALA4775663

Type: Binding

Description: Displacement of [3H]ZM2421385 from adenosine A2A receptor expressed in human HeLa cell membranes at 1 uM incubated for 30 mins by scintillation counting method

Format: BAO_0000249

Organism: Homo sapiens

Cell type: HeLa

Subcellular Fraction: Cell membrane

Target: Adenosine A2a receptor(ALA251)

Document: ALA4765483

Displacement of [3H]ZM2421385 from adenosine A2A receptor expressed in human HeLa cell membranes at 1 uM incubated for 30 mins by scintillation counting method: 1

Associated Items: Associated Bioactivities Associated Compounds

Activity Charts

Bioactivity

Activity Types for Assay ALA4775663

Inhibition

Total(165)

Compound Summary

Parent Molecular Weight	ALogP	Polar Surface Area
328.39	3.12	3.12
310.44	3.15	3.15
266.32	2.05	2.05
266.32	1.89	1.89
282.39	2.52	2.52
252.29	1.55	1.55
266.32	1.94	1.94
294.38	2.67	2.67
252.29	1.66	1.66
342.42	3.46	3.46
236.30	1.97	1.97
294.38	2.58	2.58
264.28	1.86	1.86
282.39	2.52	2.52
250.25	1.47	1.47
294.38	2.72	2.72
296.42	2.90	2.90
266.32	1.94	1.94
280.35	2.33	2.33
236.23	1.08	1.08
250.25	1.47	1.47
268.36	1.71	1.71
296.42	2.49	2.49
280.35	2.28	2.28
294.38	2.67	2.67
264.28	1.86	1.86
266.32	1.64	1.64
280.35	2.02	2.02
264.28	1.81	1.81
278.31	2.20	2.20
280.35	2.33	2.33
296.42	2.49	2.49
280.35	2.28	2.28
264.28	1.86	1.86
278.31	2.25	2.25
280.35	2.02	2.02
264.28	1.81	1.81
278.31	2.20	2.20
220.23	1.50	1.50
252.29	1.55	1.55
312.32	2.65	2.65
262.31	2.52	2.52
294.38	2.27	2.27
280.35	2.33	2.33
344.46	3.28	3.28
294.38	2.41	2.41
308.40	3.06	3.06
294.38	2.27	2.27
308.40	3.06	3.06
236.23	1.08	1.08
246.27	1.89	1.89
294.38	2.67	2.67
250.25	1.42	1.42
246.27	1.89	1.89
294.38	2.67	2.67
278.38	2.99	2.99
278.31	2.11	2.11
278.31	2.20	2.20
308.40	2.92	2.92
342.42	3.46	3.46
310.44	2.74	2.74
312.32	2.65	2.65
268.36	1.71	1.71
264.35	2.75	2.75
310.44	2.88	2.88
280.35	2.33	2.33
292.34	2.45	2.45
344.46	3.28	3.28
292.34	2.59	2.59
264.28	1.86	1.86
326.35	2.99	2.99
220.23	1.50	1.50
266.32	1.89	1.89
262.31	2.52	2.52
262.33	2.36	2.36
278.31	2.20	2.20
328.39	2.82	2.82
308.40	2.92	2.92
310.44	2.88	2.88
292.34	2.45	2.45
294.38	2.58	2.58
294.38	2.41	2.41
328.39	2.82	2.82
248.28	2.28	2.28
280.35	2.03	2.03
296.42	2.49	2.49
264.35	2.75	2.75
250.25	1.42	1.42
292.33	2.59	2.59
328.39	3.12	3.12
278.31	2.11	2.11
262.33	2.36	2.36
252.29	1.25	1.25
326.35	2.99	2.99
248.28	2.28	2.28
236.30	1.97	1.97
278.38	2.99	2.99
294.38	2.72	2.72
278.31	2.25	2.25
280.35	2.03	2.03