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Selectivity index, ratio of IC50 for displacement of Alexa Fluor 647 labelled ligand from 6His-tagged BRD4 BD1 (1 to 477 residue)/BD2 Y390A mutant (un...

Basic Information

ID: ALA4809908

Type: Binding

Description: Selectivity index, ratio of IC50 for displacement of Alexa Fluor 647 labelled ligand from 6His-tagged BRD4 BD1 (1 to 477 residue)/BD2 Y390A mutant (unknown origin) to IC50 for displacement of Alexa Fluor 647 labelled ligand from 6His-tagged BRD4 BD2 (1 to 477 residue)/BD1 Y97A mutant (unknown origin)

Format: BAO_0000019

Organism: Homo sapiens

Target:  Unchecked(ALA612545)

Document:  ALA4808200

Selectivity index, ratio of IC50 for displacement of Alexa Fluor 647 labelled ligand from 6His-tagged BRD4 BD1 (1 to 477 residue)/BD2 Y390A mutant (unknown origin) to IC50 for displacement of Alexa Fluor 647 labelled ligand from 6His-tagged BRD4 BD2 (1 to 477 residue)/BD1 Y97A mutant (unknown origin): 1

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
325.371.151.15
414.483.963.96
339.162.162.16
339.401.711.71
364.411.631.63
378.432.922.92
390.441.891.89
362.432.622.62
386.881.891.89
323.402.172.17
353.422.322.32
365.431.531.53
367.452.072.07
269.301.131.13
362.432.652.65
311.382.172.17
395.461.681.68
379.462.092.09
339.401.711.71
323.402.492.49
353.421.941.94
348.412.412.41
351.411.411.41
339.401.661.66
367.410.900.90
412.491.241.24
379.462.092.09
323.402.492.49
390.441.861.86
226.282.032.03
297.361.781.78
381.431.551.55
349.391.801.80
283.331.391.39
309.371.921.92
365.431.971.97
325.371.161.16
365.431.531.53
325.371.421.42
339.401.291.29
297.361.731.73
353.421.701.70