Basic Information
ID: ALA4810288
Type: Binding
Description: Antagonist activity at human androgen receptor expressed in HEK-293 cells harboring GRE-LUC and CMV-renilla luciferase assessed as inhibition of transactivation incubated for 24 hrs in presence of R1881 by dual luciferase assay
Organism: Homo sapiens
Cell type: HEK293
Activity Charts
Bioactivity
Activity Types for Assay ALA4810288
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 430.38 | 2.88 | 2.88 |
| 464.44 | 3.99 | 3.99 |
| 405.35 | 4.06 | 4.06 |
| 478.47 | 4.94 | 4.94 |
| 432.38 | 3.97 | 3.97 |
| 356.28 | 2.30 | 2.30 |
| 434.35 | 2.76 | 2.76 |
| 357.33 | 1.60 | 1.60 |
| 433.37 | 3.36 | 3.36 |
| 339.28 | 1.56 | 1.56 |
| 431.39 | 4.57 | 4.57 |
| 434.35 | 2.76 | 2.76 |
| 407.27 | 2.58 | 2.58 |
| 433.37 | 3.36 | 3.36 |
| 417.19 | 2.93 | 2.93 |
| 304.74 | 1.80 | 1.80 |
| 457.43 | 5.24 | 5.24 |