Basic Information
ID: ALA4810324
Type: Binding
Description: Antagonist activity at human TRPV1 expressed in CHO cells assessed as inhibition of capsaicin-induced TRPV1 activation by FLIPR method
Format: BAO_0000219
Organism: Homo sapiens
Cell type: CHO
Target: Vanilloid receptor(ALA4794)
Document: ALA4808213
Antagonist activity at human TRPV1 expressed in CHO cells assessed as inhibition of capsaicin-induced TRPV1 activation by FLIPR method: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4810324
Ki
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 516.56 | 4.27 | 4.27 |
| 409.43 | 4.33 | 4.33 |
| 427.42 | 4.47 | 4.47 |
| 427.42 | 4.47 | 4.47 |
| 441.44 | 5.03 | 5.03 |
| 507.03 | 4.75 | 4.75 |
| 518.92 | 4.48 | 4.48 |
| 411.79 | 4.54 | 4.54 |
| 439.91 | 5.41 | 5.41 |
| 446.23 | 5.20 | 5.20 |
| 416.35 | 5.34 | 5.34 |
| 434.34 | 5.47 | 5.47 |
| 443.80 | 5.24 | 5.24 |
| 441.44 | 5.03 | 5.03 |
| 460.33 | 5.50 | 5.50 |
| 457.90 | 5.55 | 5.55 |
| 428.24 | 5.06 | 5.06 |
| 462.69 | 5.71 | 5.71 |
| 409.43 | 4.33 | 4.33 |
| 460.33 | 5.50 | 5.50 |
| 429.78 | 4.68 | 4.68 |
| 428.24 | 5.06 | 5.06 |
| 460.33 | 5.50 | 5.50 |
| 450.80 | 5.99 | 5.99 |
| 417.89 | 4.96 | 4.96 |
| 443.80 | 5.24 | 5.24 |
| 477.42 | 5.35 | 5.35 |
| 442.27 | 5.62 | 5.62 |
| 460.33 | 5.50 | 5.50 |
| 446.23 | 5.20 | 5.20 |
| 427.42 | 4.47 | 4.47 |
| 443.87 | 4.99 | 4.99 |
| 443.87 | 4.99 | 4.99 |
| 411.79 | 4.54 | 4.54 |
| 491.45 | 5.91 | 5.91 |
| 441.44 | 5.03 | 5.03 |
| 417.89 | 4.96 | 4.96 |
| 476.71 | 6.27 | 6.27 |
| 479.78 | 5.56 | 5.56 |
| 425.88 | 4.85 | 4.85 |
| 423.45 | 4.90 | 4.90 |
| 429.78 | 4.68 | 4.68 |
| 448.37 | 6.04 | 6.04 |
| 429.78 | 4.68 | 4.68 |
| 443.80 | 5.24 | 5.24 |
| 474.35 | 6.06 | 6.06 |
| 443.87 | 4.99 | 4.99 |
| 481.92 | 6.40 | 6.40 |
| 434.34 | 5.47 | 5.47 |
| 429.78 | 4.68 | 4.68 |
| 428.24 | 5.06 | 5.06 |
| 446.23 | 5.20 | 5.20 |
| 446.23 | 5.20 | 5.20 |
| 441.44 | 5.03 | 5.03 |
| 462.69 | 5.71 | 5.71 |
| 427.42 | 4.47 | 4.47 |
| 460.26 | 5.76 | 5.76 |
| 476.71 | 6.27 | 6.27 |
| 450.80 | 5.99 | 5.99 |
| 467.89 | 5.84 | 5.84 |
| 425.88 | 4.85 | 4.85 |
| 439.91 | 5.41 | 5.41 |