Basic Information
ID: ALA4810626
Type: Binding
Description: Displacement of Kinase tracer 236 from biotinylated DYRK1A (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 1.5 hrs by TR-FRET assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4810626
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 302.34 | 2.95 | 2.95 |
| 212.22 | 0.77 | 0.77 |
| 226.24 | 1.23 | 1.23 |
| 316.37 | 3.26 | 3.26 |
| 294.32 | 1.17 | 1.17 |
| 270.30 | 1.26 | 1.26 |
| 253.31 | 2.10 | 2.10 |
| 239.28 | 2.09 | 2.09 |
| 240.27 | 1.25 | 1.25 |
| 254.30 | 1.56 | 1.56 |
| 266.31 | 1.78 | 1.78 |
| 254.30 | 1.56 | 1.56 |
| 241.26 | 0.65 | 0.65 |
| 254.30 | 1.56 | 1.56 |
| 309.38 | 1.33 | 1.33 |
| 254.30 | 1.56 | 1.56 |
| 239.28 | 1.86 | 1.86 |
| 336.32 | 2.97 | 2.97 |
| 284.30 | 1.73 | 1.73 |
| 239.28 | 2.09 | 2.09 |
| 280.34 | 2.03 | 2.03 |
| 270.30 | 1.26 | 1.26 |
| 294.36 | 2.56 | 2.56 |
| 322.37 | 1.80 | 1.80 |
| 280.34 | 2.03 | 2.03 |
| 322.29 | 2.57 | 2.57 |
| 294.32 | 1.02 | 1.02 |
| 239.28 | 1.86 | 1.86 |
| 294.36 | 2.42 | 2.42 |
| 319.17 | 2.01 | 2.01 |
| 280.33 | 2.17 | 2.17 |
| 258.26 | 1.39 | 1.39 |
| 308.27 | 2.27 | 2.27 |
| 306.37 | 2.42 | 2.42 |
| 282.31 | 1.28 | 1.28 |
| 312.38 | 2.05 | 2.05 |
| 253.31 | 2.10 | 2.10 |
| 239.28 | 1.86 | 1.86 |
| 240.27 | 1.25 | 1.25 |
| 366.17 | 1.86 | 1.86 |
| 284.30 | 1.73 | 1.73 |
| 294.36 | 2.57 | 2.57 |
| 236.30 | 1.67 | 1.67 |
| 274.72 | 1.91 | 1.91 |
| 284.30 | 1.73 | 1.73 |
| 280.34 | 2.03 | 2.03 |
| 298.35 | 1.66 | 1.66 |
| 296.38 | 2.81 | 2.81 |
| 240.27 | 1.25 | 1.25 |
| 270.30 | 1.26 | 1.26 |
| 231.30 | 1.99 | 1.99 |
| 282.35 | 2.38 | 2.38 |
| 278.32 | 1.64 | 1.64 |
| 270.30 | 1.26 | 1.26 |
| 239.28 | 1.86 | 1.86 |
| 254.30 | 1.56 | 1.56 |
| 252.28 | 1.40 | 1.40 |
| 274.72 | 1.91 | 1.91 |
| 266.31 | 1.79 | 1.79 |
| 281.32 | 0.72 | 0.72 |
| 281.32 | 0.72 | 0.72 |
| 254.30 | 1.56 | 1.56 |
| 230.27 | 0.91 | 0.91 |
| 307.36 | 0.98 | 0.98 |
| 267.34 | 2.58 | 2.58 |