Basic Information
ID: ALA4810633
Type: Binding
Description: Inhibition of wild-type human partial length DYRK1A (H129 to S509 residues) expressed in mammalian expression system assessed as remaining activity at 1 uM by Kinomescan method relative to control
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4810633
Activity
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 294.32 | 1.17 | 1.17 |
| 240.27 | 1.25 | 1.25 |
| 266.31 | 1.78 | 1.78 |
| 254.30 | 1.56 | 1.56 |
| 284.30 | 1.73 | 1.73 |
| 280.34 | 2.03 | 2.03 |
| 280.33 | 2.17 | 2.17 |
| 258.26 | 1.39 | 1.39 |
| 280.34 | 2.03 | 2.03 |
| 240.27 | 1.25 | 1.25 |
| 270.30 | 1.26 | 1.26 |
| 281.32 | 0.72 | 0.72 |
| 281.32 | 0.72 | 0.72 |