Assay Report Card

Basic Information

ID: ALA4813178

Type: Binding

Description: State dependent inhibition of human Nav1.5 expressed in HEK293 cells assessed as shift in compound IC50 at rested state at membrane potential of -120 mV relative to partially inactivated state at membrane potential of -95 mV

Organism: Homo sapiens

Cell type: HEK293

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
581.495.385.38