Basic Information
ID: ALA4814390
Type: Binding
Description: Inhibition of N-terminal hexahistidine-tagged human LSD1 (1 to 852 amino acids) expressed in Escherichia coli BL21 (DE3) cells using H3K4me2 peptide as substrate preincubated for 5 mins followed by substrate addition and measured for 30 mins by peroxidase-coupled method
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4814390
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 443.55 | 3.39 | 3.39 |
| 455.60 | 4.42 | 4.42 |
| 531.70 | 6.08 | 6.08 |
| 599.70 | 7.10 | 7.10 |
| 455.60 | 4.42 | 4.42 |
| 443.55 | 3.39 | 3.39 |
| 566.15 | 6.74 | 6.74 |
| 455.60 | 4.42 | 4.42 |
| 599.70 | 7.10 | 7.10 |
| 599.70 | 7.10 | 7.10 |